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Letters in Drug Design & Discovery publishes original letters on all areas of rational drug design and discovery including medicinal chemistry, in-silico drug design, combinatorial chemistry, high-throughput screening, drug targets, and structure-activity relationships. The emphasis will be on publishing quality papers very rapidly. Letters will be processed rapidly by taking full advantage of Internet technology for both the submission and review of manuscripts. The journal is essential reading to all pharmaceutical scientists involved in research in drug design and discovery.

Publisher: Bentham Science Publishers

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Volume 8, Number 2, February 2011

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Articles

Graphical Abstracts
pp. i-iv(4)
Author: Bentham Sience Publishers,

BM0701: Antibiotic Transport and Efflux: New Strategies to Combat Bacterial Resistance (ATENS)
pp. 101-101(1)
Authors: Pages, Jean-Marie; Pascu, Mihail-Lucian; Amaral, Leonard; Luisi, Ben; Hajos, Gyorgy; Fanning, Seamus; Henderson, Peter

Heterocyclic Compounds as MDR Modulators
pp. 102-113(12)
Authors: Hajos, Gyorgy; Jemnitz, Katalin; Riedl, Zsuzsanna; Takacs, Daniella; Veres, Zsuzsa

Mechanisms of Antibiotic Resistance in Salmonella: Efflux Pumps, Genetics, Quorum Sensing and Biofilm Formation
pp. 114-123(10)
Authors: Martins, Marta; McCusker, Matthew; Amaral, Leonard; Fanning, Seamus

Time Stability Studies of Quinazoline Derivative Designed to Fight Drug Resistance Acquired by Bacteria
pp. 124-129(6)
Authors: Militaru, Andra; Smarandache, Adriana; Mahamoud, Abdallah; Alibert, Sandrine; Pages, Jean-Marie; Pascu, Mihail-Lucian

Thioridazine: Alternative and Potentially Effective Therapy of the XDRTB Patient
pp. 130-132(3)
Authors: Amaral, Leonard; Martins, Marta; Viveiros, Miguel

Quorum Sensing Inhibition by Phenothiazines and Related Compounds
pp. 133-137(5)
Authors: Gabor Varga, Zoltan; Agnes Szabo, Mira; Schelz, Zsuzsanna; Szegedi, Erno; Amaral, Leonard; Molnar, Jozsef

Synthesis and Comparison of the Antitumor Activities of Steroids on ABCB1-transfected Mouse Lymphoma and Human Ovary Carcinoma
pp. 138-147(10)
Authors: Serly, Julianna; Vincze, Iren; Somlai, Csaba; Hodoniczki, Laszlo; Molnar, Jozsef

Expression of P-gp, MRP, LRP, GST-π and TopoIIα and Acquired Resistance to Cisplatin in Human Lung Adenocarcinoma Cells
pp. 148-153(6)
Authors: Wang, Jiarui; He, Zhongzhou; Zhang, Lichuan; Li, Encheng; Meng, Qiang; Zou, Lijuan; Molnar, Joseph; Wang, Qi

Synthesis and Biological Evaluation of Gemfibrozil Chiral Analogues as Potential PPARα Agonists
pp. 154-158(5)
Authors: De Filippis, Barbara; Giampietro, Letizia; Giancristofaro, Antonella; Ammazzalorso, Alessandra; Fantacuzzi, Marialuigia; Maccallini, Cristina; Petruzzelli, Michele; Amoroso, Rosa

Integrated Web-Based ab initio Modeling Platform for G-protein Coupled Receptors
pp. 159-171(13)
Authors: Subramanian, Govindan; Sud, Manish; Billakanti, Sam; Laoui, Adel

Search of QSAR Models for Predicting the Antiprotozoal Activity and Cytotoxicity In Vitro of a Group of Pentamidine Analogous Compounds
pp. 172-180(9)
Authors: Garcia-Domenech, Ramon; Denise Manhenje, Isabel; Monje, Yamileth; Lopez-Gonzalez, Adassa; Marco, Rafael; Tacho, Catalina; Galvez, Jorge

The Global Component-Target Network in Panax Ginseng C
pp. 181-188(8)
Authors: Zhang, Fan; Li, Chun-Yang; Wang, En-Qin; Li, Wen-Wen; Yu, Qi-Jia; Wen, Xin; Liu, Jun-Jie; Bao, Jin-Ku

Synthesis and Biological Evaluation of Some [1,2,4]Triazolo[3,4-b][1,3,4]Thiadiazoles and [1,2,4]Triazolo[3,4-b][1,3,4]Thiadiazines
pp. 189-200(12)
Authors: Shankara Naveena, Channamata; Poojary, Boja; Chandrashekhar, Chikkanna; Suchetha Kumari, Nalilu

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