Letters in Drug Design & Discovery

The Anticancer Activity of the N-Terminal CARD-Like Domain of Arginine Deiminase (ADI) from Pseudomonas aeruginosa
pp. 403-412(10)
Authors: Kundu, Madhuchhanda; Thomas, Johnson; Fialho, Arsenio M.; Kwan, Jennifer M.; Moreira, Leonilde M.; Mahfouz, Magdy; Das Gupta, Tapas K.; Chakrabarty, Ananda M.

Synthesis and Evaluation of Anthelmintic and Cytotoxic Properties of [2,5']Bis-1,3-Azole Analogs of Bengazoles
pp. 413-419(7)
Authors: Scarone, Laura; Fajardo, Jose; Saldana, Jenny; Dominguez, Laura; Esposito, Pablo; Demastteis, Sylvia; Wipf, Peter; Manta, Eduardo; Serra, Gloria

The Synthesis and Activity Evaluation of a Bestatin Derivative (LYP) as an Aminopeptidase N Inhibitor
pp. 420-423(4)
Authors: Luan, Yepeng; Wang, Xuejian; Zhu, Huawei; Qu, Xianjun; Fang, Hao; Xu, Wenfang

Synthesis and Bioactivities of 2-Azetidinones as Cholesterol Absorption Inhibitors
pp. 424-427(4)
Authors: Ji, Jianfeng; Zhao, Rui; Huang, Wenlong; Zhang, Huibin; Zhou, Jinpei; Wang, Yubin; Qian, Hai

Multivariate Linear Regression Models Based on ADME Descriptors and Predictions of ADMET Profile for Structurally Diverse Thermolysin Inhibitors
pp. 428-436(9)
Authors: Khan, Mahmud T.H.; Sylte, Ingebrigt

Anti-Amyloid Effects of Small Molecule Aβ-Binding Agents in PS1/APP Mice
pp. 437-444(8)
Authors: Cohen, A. D.; Ikonomovic, M. D.; Abrahamson, E. E.; Paljug, W. R.; DeKosky, S. T.; Lefterov, I. M.; Koldamova, R. P.; Shao, L.; Debnath, M. L.; Mason, N. S.; Mathis, C. A.; Klunk, W. E.

Synthesis and Pharmacological Activity of Thiourea Derivatives of 1,7,8,9-Tetramethyl-4-azatricyclo[5.2.1.02,6]dec-8-ene-3,5-dione
pp. 445-450(6)
Authors: Struga, Marta; Kossakowski, Jerzy; Koziol, Anna E.; Lis, Tateusz; Kedzierska, Ewa; Fidecka, Sylwia

Synthesis, Spectral Studies and Anti-Bacterial Activity of Novel Substituted aryl/heteroaryl-(12-substituted phenyl-12H-7-oxa-8, 10-diazabenzo[ a]anthracen-11-yl)-amine
pp. 451-455(5)
Authors: Mahammed, K. A.; Venugopala, K. N.; Arunachalam, P. N.; Raju, K. M.

Anticonvulsant Activity of A Novel Series of 2,5-Disubstituted 1,3,4-Oxadiazoles: Semicarbazones Based Pharmacophoric Model Studies
pp. 456-463(8)
Authors: Rajak, Harish; Veerasamy, Ravichandran; Singour, Pradeep; Kharya, Murli D.; Mishra, Pradeep

8-(Trifluoromethyl)-1,2,3,4,5-benzopentathiepin-6-amine: Novel Aminobenzopentathiepine having In Vivo Anticonvulsant and Anxiolytic Activities
pp. 464-467(4)
Authors: Khomenko, Tatyana M.; Tolstikova, Tatyana G.; Bolkunov, Alexey V.; Dolgikh, Margarita P.; Pavlova, Alla V.; Korchagina, Dina V.; Volcho, Konstantin P.; Salakhutdinov, Nariman F.

Synthesis and Structure-Activity Relationship Study of 2-Substituted- 5-(5-nitro-2-thienyl)-1,3,4-thiadiazoles as Anti-Helicobacter pylori Agents
pp. 468-474(7)
Authors: Foroumadi, Alireza; Sedaghat, Somayeh; Emami, Saeed; Yazdanian, Maryam; Moshafi, Mohammad H.; Safavi, Maliheh; Sakhteman, Amirhossein; Firoozpour, Loghman; Vosooghi, Mohsen; Shafiee, Abbas