Letters in Drug Design & Discovery

Synthesis of 4-substituted-3-hydroxy-5-oxo-10-oxa-4-azatricyclo[5.2.1]dec- 3-yl Acetic Acid Ethyl Esters as Norcantharidin Analogues
pp. 1-7(7)
Authors: Sauer, Benjamin; Gilbert, Jayne; Sakoff, Jennette A.; McCluskey, Adam

Involvement of Serotonin in the Acute Dependence Produced by μ, and K Opioid Agonists
pp. 8-12(5)
Author: Capasso, Anna

Buprenorphine and Methadone Maintenance Treatment - Sexual Behaviour and Dysfunction Prevalence
pp. 13-13(1)
Authors: Giacomuzzi, S. M.; Khreis, A.; Riemer, Y.; Garber, K.; Ertl, M.

Computer-Aided Drug Design for Cancer-Causing H-Ras p21 Mutant Protein
pp. 14-20(7)
Authors: Jayakanthan, Mannu; Wadhwa, Gulshan; Mohan, Thangavel M.; Arul, Loganathan; Balasubramanian, Ponnusamy; Sundar, Durai

Synthesis, Antibacterial Activity of 2,4-Disubstituted Oxazoles and Thiazoles as Bioisosteres
pp. 21-28(8)
Authors: Kaspady, Mohamed; Narayanaswamy, Venugopala K.; Raju, Mohana; Rao, Gopal K.r.i.s.h.n.a.

Identification of GCP II Inhibitors Based on 4-Arylmethyl-3-(4- carboxyphenyl)-5-hydroxyisoxazole Scaffold
pp. 29-32(4)
Authors: Teus, M.; Jirgensons, A.; Dambrova, M.; Mezhapuke, R.; Parsons, C. G.; Danysz, W.

Structural and Morphological Studies of Cationic Liposomes-DNA Complexes
pp. 33-37(5)
Authors: Sun, Yan; Migueliz, Itziar; Navarro, Gemma; de Ilarduya, Conchita T.

Pharmacophore Searching of Benzofuran Derivatives for Selective CYP19 Aromatase Inhibition
pp. 38-45(8)
Authors: Nagar, Shuchi; Islam, Md A.; Das, Suvadra; Mukherjee, Arup; Saha, Achintya

Evaluation of In-Vivo Anti-Implantation and In-Vitro Anti-Proliferative Activities of Substituted 3-phenyl-4-phenylvinyl Benzopyranone Derivatives
pp. 46-50(5)
Authors: Gupta, Atul; Sharma, Ramesh; Balapure, Anil K.; Keshri, Govind; Singh, M. M.; Ray, Suprabhat

Synthesis and Antitumor Activity of Novel 4-Chloro-3-Arylmaleimide Derivatives
pp. 51-55(5)
Authors: Xu, Guiqing; He, Qiaojun; Yang, Bo; Hu, Yongzhou

DNA Binders: 1. Evaluation of DNA-Interactive Ability, Design, and Synthesis of Novel Intercalating Agents
pp. 56-62(7)
Authors: Sechi, Mario; Derudas, Marco; Dallocchio, Roberto; Dessì, Alessandro; Cosseddu, Alessia; Paglietti, Giuseppe

Susceptibility of Staphylococcus spp. Isolated from Milk of Goats with Mastitis to Antibiotics and Green Propolis Extracts
pp. 63-68(6)
Authors: Santos Neto, T. M.; Mota, R. A.; Silva, L. B.G.; Viana, D. A.; Lima-Filho, J. L.; Sarubbo, L. A.; Converti, A.; Porto, A. L.F.

Synthesis and Antibacterial and Antifungal Activity of 5-Substituted Imidazolones
pp. 69-77(9)
Authors: Khan, Khalid M.; Mughal, Uzma R.a.s.o.o.l.; Khan, Sadia; Khan, Saira; Perveen, Shahnaz; Choudhary, M. I.q.b.a.l.

Solution-Phase Parallel Synthesis of N-Arylisoquinuclidines
pp. 78-81(4)
Authors: Borne, Ronald F.; Levi, Mark S.; Faruk Khan, M. O.; Wilson, Norman H.

Development of an Economical, Single Step Synthesis of FAZA, a Clinical Hypoxia Marker, and Potential Synthons to Prepare its Positional Analogs
pp. 82-85(4)
Authors: Kumar, P.; Emami, S.; McEwan, A. J.B.; Wiebe, L. I.