Letters in Drug Design & Discovery

Synthesis, DNA-Binding Ability and Biological Activity of C8 Linked G1 Dendrimer-Pyrrolobenzodiazepine Conjugates as Anticancer Agents
pp. 424-432(9)
Authors: Kamal, Ahmed; Balakishan, G.; Rajender,; Sreekanth, K.; Reddy, D. R.; Reddy, M. K.a.s.h.i.; Sen, Subrata; Kurian, Nisha; Juvekar, Aarti S.; Zingde, Surekha M.

Sesquiterpene Lactones and their Anti-Tumor Activity from the Flowers of Inula Britannica
pp. 433-436(4)
Authors: Qi, Jin-Long; Fu, Yan; Shi, Xiao-Wei; Wu, Yi-Bing; Wang, Yun-Zhi; Zhang, Di-Qun; Shi, Qing-Wen

3D-QSAR Studies of Various Diaryl Urea Derivatives of Multi-targeted Receptor Tyrosine Kinase Inhibitors: Molecular Field Analysis Approach
pp. 437-448(12)
Authors: Kansal, Neha; Silakari, Om; Ravikumar, Muttineni

3D-QSAR Analysis on N-Phenylacetanoyl-L-Homoserine Lactones as Inhibitors of Bacterial Quorum Sensing via CoMFA Approach
pp. 449-453(5)
Authors: Sun, Ping-Hua; Yang, Zhao-Qi; Chen, Wei-Min; Liu, Qian; Yao, Xin-Sheng

Synthesis and In Vitro Antiproliferative Activity of Diphenyl(piperidin-4- yl)thioamide Methanol Derivatives
pp. 454-461(8)
Authors: Benaka Prasad, Salekoppal B.; Vinaya, Mallappanahally K.a.m.b.a.p.p.a.; Ananda Kumar, Channapille K.S.; Swarup, Sanjay; Rangappa, Kanchugarakoppal S.u.b.b.e.g.o.w.d.a.

Release of a Poorly Soluble Drug from Cross-Linked β-Cyclodextrin-Based Polymer Pellets Prepared via Extrusion/Spheronisation
pp. 462-470(9)
Authors: Bon, Pierre; Joudieh, Samer; Lahiani-Skiba, Malika; Bounoure, Frederic; Dechelotte, Pierre; Skiba, Mohamed

96-Well Plate Surface Tension Measurements for Fast Determination of Drug Solubility
pp. 471-476(6)
Authors: Heikkila, Tiina; Peltonen, Leena; Taskinen, Saila; Laaksonen, Timo; Hirvonen, Jouni