Letters in Drug Design & Discovery

Evaluation of the Ability of an Organic Derivative of Ruthenium(II) to Reinforce the Cytotoxicity of Fast Neutron Against Malignant Cells in Culture
pp. 1-6(6)
Authors: Bischoff, P.; Leyva, L.; Malek, F.; Benzina, S.; Denis, J. M.; Gueulette, J.; Dufour, P.; Gaiddon, C.; Loeffler, J. P.; Sirlin, C.; Pfeffer, M.

CoMFA Study, Syntheses, Antitubercular and Anticancer Activity of Some Novel 1,4-Dihydropyridines
pp. 7-14(8)
Authors: Kumar, B.R. P.; Yuvaraj, S.; Srivastava, Anil; Chaturvedi, Vanitha; Manju, Y. K.; Suresh, B.; Nanjan, M. J.

Synthesis, In Vitro Evaluations and Structure-Activity Assessment of Pyrrole Hydrazones as Potential Tuberculostatics
pp. 15-24(10)
Author: Bijev, A.

Synthesis and Evaluation of N-Aryl 2-Aminothiazole-4-Carboxamide Derivatives for Activity Against TB
pp. 25-28(4)
Authors: Riggs, R. M.; Jennings, R. K.; Derstine, E. R.; Nguyen, T. M.; Trinh, T.; Riordan, J. M.

Immunomodulation and Anti-Inflammatory Effects of Macrolides: Old Drugs with Fascinating New Perspectives
pp. 29-35(7)
Author: Starakis, I.

Selective Inhibition of Neuronal Nitric Oxide Synthase by L-Arginine Derivatives
pp. 36-38(3)
Authors: Capasso, Anna; Saturnino, Carmela; Buonerba, Mariafrancesca

Design and Synthesis of 2-Azetidinone Cholesterol Absorption Inhibitors
pp. 39-42(4)
Authors: Zhang, Huibin; Wang, Yubin; Zhao, Rui; Huang, Wenlong; Li, Yunman; Zhou, Jinpei

Solution Phase Synthesis of a 3,5,7-Substituted Indolin-2-one Library as Potential CDK2 Inhibitor Isosteres
pp. 43-47(5)
Authors: Tymoshenko, Dmytro O.; Gregg, Brian T.; Hirsch, Matthew J.; Butcher, Jennifer L.

Inhibition of 17β -Hydroxysteroid Dehydrogenase (17β -HSD) by Imidazole-Based Compounds
pp. 48-51(4)
Authors: Ahmed, Sabbir; Olusanjo, Moniola S.; Shahid, Imran; Owen, Caroline P.

Synthesis and Chymotrypsin Inhibitory Activity of Substituted Oxazolones
pp. 52-56(5)
Authors: Khan, Khalid M.; Mughal, Uzma R.a.s.o.o.l.; Lodhi, Muhammad A.r.i.f.; Choudhary, Muhammad I.q.b.a.l.

Classical and Fragment-Based Hologram Structure-Activity Relationships for a Series of Analgesic Cyclic Imides
pp. 57-64(8)
Authors: Andricopulo, A. D.; Borchhardt, D. M.; Castilho, M. S.

Central Administration of L-Ser-L-His and L-Ile-L-His Induced Sedative Effects Under an Acute Stressful Condition in Chicks
pp. 65-68(4)
Authors: Furuse, Mitsuhiro; Tsuneyoshi, Yousuke; Tomonaga, Shozo; Yamane, Haruka; Morishita, Koji; Denbow, D. M.

Flavylium Salts as Precursors of Biologically Active Chalcones
pp. 69-73(5)
Authors: Werbovetz, Karl A.; George, Tesmol G.; Richard, Julian; Barszcz, Todd; Capers, Jeffrey

Antifungal Activity of Goniothalamin Enantiomers
pp. 74-78(5)
Authors: Fatima, Angelo d.; Martins, Cleide Viviane B.u.z.a.n.e.l.l.o.; de Resende, Maria A.p.a.r.e.c.i.d.a.; Ferreira Magalhaes, Thais F.u.r.t.a.d.o.; Santiago Lima, Bruno H.e.n.r.i.q.u.e.; Watanabe, Gisele A.l.m.e.i.d.a.; Gois Ruiz, Ana L.T.; de Carvalho, Joao E.r.n.e.s.t.o.; Pilli, Ronaldo A.l.o.i.s.e.