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Letters in Drug Design & Discovery publishes original letters on all areas of rational drug design and discovery including medicinal chemistry, in-silico drug design, combinatorial chemistry, high-throughput screening, drug targets, and structure-activity relationships. The emphasis will be on publishing quality papers very rapidly. Letters will be processed rapidly by taking full advantage of Internet technology for both the submission and review of manuscripts. The journal is essential reading to all pharmaceutical scientists involved in research in drug design and discovery.

Publisher: Bentham Science Publishers

Volume 4, Number 6, September 2007
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Articles

Inhibition of Human Leucocyte Elastase by Novel Thieno-1,3-oxazin-4-ones and Thieno-1,3-thioxazin-4-ones
pp. 386-393(8)
Authors: N.A. Santagati,; L. Salerno,; C. Di Giacomo,; L. Vanella,; S. Ronsisvalle,

Inhibition of Human Leucocyte Elastase by Novel Thieno-1,3-oxazin-4-ones and Thieno-1,3-thioxazin-4-ones
pp. 386-393(8)
Authors: N.A. Santagati,; L. Salerno,; C. Di Giacomo,; L. Vanella,; S. Ronsisvalle,

Synthesis and In Vitro Biochemical Evaluation of a Series of Compounds as Potential Inhibitors of Estrone Sulfatase (ES) and the Role of pKa in both the Synthesis and the Inhibitory Activity of the Potential Inhibitors
pp. 394-398(5)
Authors: Caroline P. Owen,; Mijal Patel,; Chirag K Patel,; Tim Cartledge,; Sabbir Ahmed,

Synthesis and In Vitro Biochemical Evaluation of a Series of Compounds as Potential Inhibitors of Estrone Sulfatase (ES) and the Role of pKa in both the Synthesis and the Inhibitory Activity of the Potential Inhibitors
pp. 394-398(5)
Authors: Caroline P. Owen,; Mijal Patel,; Chirag K Patel,; Tim Cartledge,; Sabbir Ahmed,

Synthesis and In Vitro Biochemical Evaluation of a Series of Cycloalkyl Esters of 4-Sulfamoylated Benzoic Acid as Inhibitors of Estrone Sulfatase (ES)
pp. 399-403(5)
Authors: Caroline P. Owen,; Chirag K. Patel,; Tim Cartledge,; Sabbir Ahmed,

Synthesis and In Vitro Biochemical Evaluation of a Series of Cycloalkyl Esters of 4-Sulfamoylated Benzoic Acid as Inhibitors of Estrone Sulfatase (ES)
pp. 399-403(5)
Authors: Caroline P. Owen,; Chirag K. Patel,; Tim Cartledge,; Sabbir Ahmed,

Synthesis and Anti-HSV-1 Activity of 1,4-dihydro-4-oxoquinoline Ribonucleosides
pp. 404-409(6)
Authors: Carla Veronica B. dos S. Canuto,; Claudia R. B. Gomes,; Isakelly P. Marques,; Leticia V. Faro,; Fernanda da Costa Santos,; Izabel Christina de P. P. Frugulhetti,; Thiago M. L. e Souza,; Anna C.Cunha,; Gilberto A. Romeiro,; Vitor F. Ferreira,; Maria Cecilia B.V.de Souza,

Synthesis and Anti-HSV-1 Activity of 1,4-dihydro-4-oxoquinoline Ribonucleosides
pp. 404-409(6)
Authors: Carla Veronica B. dos S. Canuto,; Claudia R. B. Gomes,; Isakelly P. Marques,; Leticia V. Faro,; Fernanda da Costa Santos,; Izabel Christina de P. P. Frugulhetti,; Thiago M. L. e Souza,; Anna C.Cunha,; Gilberto A. Romeiro,; Vitor F. Ferreira,; Maria Cecilia B.V.de Souza,

Classification and Prediction of Tripeptides Inhibiting HIV-1 Tat/TAR-RNA Interaction Using a Self-Organizing Map
pp. 410-416(7)
Authors: A. Givehchi,; V. Ludwig,; O. Boden,; A. Krebs,; U. Scheffer,; M. Gobel,; G. Schneider,

Classification and Prediction of Tripeptides Inhibiting HIV-1 Tat/TAR-RNA Interaction Using a Self-Organizing Map
pp. 410-416(7)
Authors: A. Givehchi,; V. Ludwig,; O. Boden,; A. Krebs,; U. Scheffer,; M. Gobel,; G. Schneider,

Structure-Based Quantitative Structure Activity Relationship Analysis of Omuralide Analogs in the 20S Proteasome: A Covalent Inhibitor COMBINE Study
pp. 417-421(5)
Authors: Jenna L. Wang,; Apurba Datta,; Gerald H. Lushington,

Structure-Based Quantitative Structure Activity Relationship Analysis of Omuralide Analogs in the 20S Proteasome: A Covalent Inhibitor COMBINE Study
pp. 417-421(5)
Authors: Jenna L. Wang,; Apurba Datta,; Gerald H. Lushington,

The Molecular Basis of COX-2 Versus COX-1 Selectivity of Lumiracoxib by Molecular Docking Studies
pp. 422-425(4)
Authors: Celia M. Correa,; Andre F. de Paula,; Gilberto M.S. da Silva,; Carlos M.R. Sant'Anna,; Carlos A. M. Fraga,; Eliezer J. Barreiro,

The Molecular Basis of COX-2 Versus COX-1 Selectivity of Lumiracoxib by Molecular Docking Studies
pp. 422-425(4)
Authors: Celia M. Correa,; Andre F. de Paula,; Gilberto M.S. da Silva,; Carlos M.R. Sant'Anna,; Carlos A. M. Fraga,; Eliezer J. Barreiro,

A Cationic Liposomal Vincristine Formulation with Improved Vincristine Retention, Extended Circulation Lifetime and Increased Anti-Tumor Activity
pp. 426-433(8)
Authors: Murray S. Webb,; Nancy L. Boman,; Dana Masin,; Donald Yapp,; Euan Ramsay,; Gigi N.C. Chiu,; Pieter R. Cullis,; Marcel B. Bally,

A Cationic Liposomal Vincristine Formulation with Improved Vincristine Retention, Extended Circulation Lifetime and Increased Anti-Tumor Activity
pp. 426-433(8)
Authors: Murray S. Webb,; Nancy L. Boman,; Dana Masin,; Donald Yapp,; Euan Ramsay,; Gigi N.C. Chiu,; Pieter R. Cullis,; Marcel B. Bally,

Isoform-Selective Regulation of Adenylyl Cyclase by Forskolin Derivatives:Prediction of Selectivity by Computer-Based Analysis
pp. 434-441(8)
Authors: Haruki Eguchi,; Kousaku Iwatsubo,; Yoshihiro Ishikawa,

Isoform-Selective Regulation of Adenylyl Cyclase by Forskolin Derivatives:Prediction of Selectivity by Computer-Based Analysis
pp. 434-441(8)
Authors: Haruki Eguchi,; Kousaku Iwatsubo,; Yoshihiro Ishikawa,

Preparation and Biological Activities of Heteroarotinoids
pp. 442-445(4)
Authors: Akimori Wada,; Yukari Mizuguchi,; Hiromi Miyake,; Miki Niihara,; Masayoshi Ito,; Kimie Nakagawa,; Toshio Okano,

Preparation and Biological Activities of Heteroarotinoids
pp. 442-445(4)
Authors: Akimori Wada,; Yukari Mizuguchi,; Hiromi Miyake,; Miki Niihara,; Masayoshi Ito,; Kimie Nakagawa,; Toshio Okano,

Lamotrigine as an Effective Treatment for Behavioral Disorders
pp. 446-452(7)
Authors: Rita Moretti,; Paola Torre,; Cristina Vilotti,; Rodolfo M. Antonello,

Lamotrigine as an Effective Treatment for Behavioral Disorders
pp. 446-452(7)
Authors: Rita Moretti,; Paola Torre,; Cristina Vilotti,; Rodolfo M. Antonello,

Release Kinetics of Ampicillin, Biocompatibility Tests with a Fibroblast Strain of a Zirconia Gel Glass
pp. 453-459(7)
Authors: M. Catauro,; M.G. Raucci,; M.A. Continenza,

Release Kinetics of Ampicillin, Biocompatibility Tests with a Fibroblast Strain of a Zirconia Gel Glass
pp. 453-459(7)
Authors: M. Catauro,; M.G. Raucci,; M.A. Continenza,

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