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Letters in Drug Design & Discovery publishes original letters on all areas of rational drug design and discovery including medicinal chemistry, in-silico drug design, combinatorial chemistry, high-throughput screening, drug targets, and structure-activity relationships. The emphasis will be on publishing quality papers very rapidly. Letters will be processed rapidly by taking full advantage of Internet technology for both the submission and review of manuscripts. The journal is essential reading to all pharmaceutical scientists involved in research in drug design and discovery.

Publisher: Bentham Science Publishers

Volume 3, Number 5, July 2006
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Articles

Quality Initiatives in Drug Discovery: Swim Don't Sink
pp. 286-288(3)
Authors: Volsen, S. G.; Parry, M. G.; Masson, M.

Design and Discovery of Novel, Potent Pyrazinone-Based Thrombin Inhibitors with a Solubilizing Amino P1-P2-Linker
pp. 289-292(4)
Authors: Bulat, S.; Bosio, S.; Papadopoulos, M. A.; Cerezo-Galvez, S.; Grabowski, E.; Rosenbaum, C.; Matassa, V. G.; Ott, I.; Metz, G.; Schamberger, J.; Sekul, R.; Feurer, A.

Target Structure-based Modeling of the Glutamate Transporter Pharmacophore
pp. 293-297(5)
Authors: Simon, A.; Bencsura, A.; Kardos, J.

Novel Benzimidazole Derivatives as Selective CB2 Inverse Agonists
pp. 298-303(6)
Authors: Page, D.; Brochu, M.-C.; Yang, H.; Brown, W.; St-Onge, S.; Martin, E.; Salois, D.

Design, Synthesis and Biological Evaluation of Novel Curcumin Analogues as Anti-Neoplastic Agents
pp. 304-310(7)
Authors: Jha, Amitabh; Zhao, Jin; Stanley Cameron, T.; De Clercq, Erik; Balzarini, Jan; Manavathu, Elias K.; Stables, James P.

Synthesis of Piperazinephen-1-ylethylamines as Potent and Selective Antagonists of the Human Melanocortin-4 Receptor
pp. 311-315(5)
Authors: Tucci, Fabio C.; Tran, Joe A.; Jiang, Wanlong; Pontillo, Joseph; Marinkovic, Dragan; White, Nicole S.; Arellano, Melissa; Fleck, Beth A.; Wen, Jenny; Saunders, John; Foster, Alan C.; Chen, Chen

Cytotoxic and COX-2 Inhibition Properties of Hydroxycinnamic Derivatives
pp. 316-320(5)
Authors: M. Marques, M. Paula; Borges, Fernanda; Sousa, Joana; Calheiros, Rita; Garrido, Jorge; Gaspar, Alexandra; Diniz, Carmen; Fresco, Paula

Lamotrigine Pharmacokinetics During Anticonception and Pregnancy
pp. 321-322(2)
Author: Sabers, A.

The NK-1 Receptor is Involved in the Antitumoural Action of L-733,060 and in the Mitogenic Action of Substance P on Human Pancreatic Cancer Cell Lines
pp. 323-329(7)
Authors: Munoz, Miguel; Rosso, Marisa; Covenas, Rafael

Synthesis and Radiopharmacological Characterisation of 86Y- and 68Ga-Labelled L-RNA Oligonucleotides as Molecular Probes for Positron Emission Tomography (PET)
pp. 330-335(6)
Authors: Schlesinger, Joern; Bergmann, Ralf; Klussmann, Sven; Wuest, Frank

Design, Synthesis and Initial In Vitro Evaluation of Novel Prodrugs for the Treatment of Cystinosis
pp. 336-345(10)
Authors: Anderson, R. J.; Cairns, D.; Cardwell, W. A.; Case, M.; Groundwater, P. W.; Hall, A. G.; Hogarth, L.; Jones, A. L.; Meth-Cohn, O.; Suryadevara, P.

The Cardiovascular Properties of Some Amide Derivatives of Pyrimidin-8-on[2,1-f]theophylline-9- Alkylcarboxylic Acids
pp. 346-350(5)
Authors: Zagorska, A.; Fhid, O.; Pawlowski, M.; Filipek, B.; Zygmunt, M.

Homocysteine and Folate Therapy in Dialysis Patients
pp. 351-355(5)
Author: Righetti, Marco

Erratum
pp. 356-356(1)

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