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Letters in Drug Design & Discovery publishes original letters on all areas of rational drug design and discovery including medicinal chemistry, in-silico drug design, combinatorial chemistry, high-throughput screening, drug targets, and structure-activity relationships. The emphasis will be on publishing quality papers very rapidly. Letters will be processed rapidly by taking full advantage of Internet technology for both the submission and review of manuscripts. The journal is essential reading to all pharmaceutical scientists involved in research in drug design and discovery.

Publisher: Bentham Science Publishers

Volume 2, Number 8, December 2005
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Review article

Rational Design of the New Antihypertensive I1-Receptor Ligand 2-(2- Biphenyl-2-yl-1-methyl-ethyl)-4,5-dihydro-1H-imidazole
pp. 571-578(8)
Authors: F. Gentili,; P. Bousquet,; A. Carrieri,; J. Feldman,; F. Ghelfi,; M. Giannella,; A. Piergentili,; W. Quaglia,; C. Vesprini,; M. Pigini,

Docking Study, Synthesis and SAH-Hydrolase Inhibitory Activity of LAdeninylalanine and Related Analogues
pp. 579-583(5)
Authors: Floquet, Nicolas; Leroy, Samuel; Muzard, Murielle; Guillerm, Georges; Behr, Jean-Bernard

Anti-tumour Activity of Some Polydentate N-Ligands: N,N-bis-(3- Substituted-5-Methylpyrazol-1yl Methyl) Arylamines and N,N,N',N'-Tetra- [(3-Substituted-5-Methylpyrazol-1yl] Para-Phenylenediamines
pp. 584-589(6)
Authors: Hadda, T. B.; Kotchevar, A. T.; Daoudi, M.; Bennani, B.; Larbi, N. B.; Kerbal, A.

Discovery of Thrombin Inhibitor Fragments from Chemical Microarray Screening
pp. 590-594(5)
Authors: Neumann, Thomas; Junker, Hans-Dieter; Keil, Oliver; Burkert, Klaus; Ottleben, Holger; Gamer, Jurgen; Sekul, Renate; Deppe, Holger; Feurer, Achim; Tomandl, Dirk; Metz, Gunther

Identification of Privileged Scaffolds from a Diversified Chemical Library forβ-Secretase Inhibition
pp. 595-600(6)
Authors: Pietrancosta, Nicolas; Quelever, Gilles; Garino, Cedrik; Laras, Younes; Burlet, Stephane; Kraus, Jean-Louis

Synthesis and Biological Evaluation of 1,2,4-Triazolo[2,3-a]pyrrole Derivatives as Alpha-4 ( α4) Integrin Antagonists
pp. 601-605(5)
Authors: Lawson, Edward C.; Kinney, William A.; Santulli, Rosemary J.; Fisher, Carol M.; Damiano, Bruce P.; Maryanoff, Bruce E.

Szeged Index - Applications for Drug Modeling#
pp. 606-624(19)
Authors: Khadikar, Padmakar V.; Karmarkar, Sneha; Agrawal, Vijay K.; Singh, Jyoti; Shrivastava, Anjali; Lukovits, Istvan; Diudea, Mircea V.

Initial Structure-Activity Relationships for a Caprolactam-based Series of Neutral Factor Xa Inhibitors: Lead Identification
pp. 625-630(6)
Authors: Bisacchi, Gregory S.; Stein, Philip D.; Gougoutas, Jack Z.; Hartl, Karen S.; Lawrence, R. M.; Liu, Eddie; Pudzianowski, Andrew; Schumacher, William A.; Sitkoff, Doree; Steinbacher, Thomas E.; Sutton, James; Zhang, Zhaoxiao; M. Seiler, Steven

Synthesis and Evaluation of p-Nitrophenylβ-D-Glucopyranosiduronic Analogues as New Triggers for β-Glucuronidase Mediated Prodrug Mono- Therapy
pp. 631-637(7)
Authors: Combaud, Damien; Thomas, Mickael; Papot, Sebastien; Gesson, Jean-Pierre

Structure Based Design of Inhibitors of Aspartic Protease of HIV-1
pp. 638-646(9)
Authors: Frecer, V.; Jedinak, A.; Tossi, A.; Berti, F.; Benedetti, F.; Romeo, D.; Miertus, S.

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