Recent Advances in the Rationale Design of GPER Ligands
Keywords: GPCRs; GPR30/GPER; agonists/antagonists; antiestrogens; atomic structures; binding modes; estrogens; homology modelling; receptor; small molecules ligands; virtual screening; “in silico” docking simulations
Document Type: Research Article
Publication date: 2012-12-01
- Current Medicinal Chemistry covers all the latest and outstanding developments in medicinal chemistry and rational drug design. Each issue contains a series of timely in-depth reviews written by leaders in the field covering a range of the current topics in medicinal chemistry. Current Medicinal Chemistry is an essential journal for every medicinal chemist who wishes to be kept informed and up-to-date with the latest and most important developments.