Macrocyclic G-Quadruplex Ligands
Keywords: Anticancer therapeutics; BCL-2; Corroles; DNA; FRET Tm; G-quadruplex; HeLa cells; Hoogsteen base pairing; SPR; Streptomyces anulatus; Telomeres; WO 0024747; WO 2004078764; antitumor; c-KIT sequence; c-MYC; cancer; cell line; cytotoxic; drug discovery; guanine; hexaoxazoles; hybrid; isoindole; leukemia; ligands; macrocycles; macrocyclic; nucleic acid; oncogenes; p-p stacking; phosphate backbone; porphyrin; porphyrins; pyrrole; telomerase-negative Saos-2 cells; telomere repeat amplification protocol (TRAP) assay; telomeric sequences; telomestatin; topology; tumor xenografts
Document Type: Research Article
Publication date: 2010-10-01
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