Journal of Enzyme Inhibition and Medicinal Chemistry

Chemical constituents of Polygala tenuifolia roots and their inhibitory activity on lipopolysaccharide-induced nitric oxide production in BV2 microglia
pp. 1-4(4)
Authors: Cho, Namki; Huh, Jungmoo; Yang, Heejung; Jeong, Eun Ju; Kim, Young Choong; Kim, Jinwoong; Sung, Sang Hyun

A screening assay for neuraminidase inhibitors using neuraminidases N1 and N3 from a baculovirus expression system
pp. 5-11(7)
Authors: Kongkamnerd, Jarinrat; Milani, Adelaide; Cattoli, Giovanni; Terregino, Calogero; Capua, Ilaria; Beneduce, Luca; Gallotta, Andrea; Pengo, Paolo; Fassina, Giorgio; Miertus, Stanislav; De-Eknamkul, Wanchai

Oxidases and oxygenases in regulation of neutrophil redox pathways in Behçet's disease patients
pp. 12-17(6)
Authors: Melikoglu, Meltem A.; Kacar, Cahit; Cort, Aysegul; Yucel, Gultekin; Aslan, Mutay

In vitro effects of some drugs on human erythrocyte glutathione reductase
pp. 18-23(6)
Authors: Karaman, Muhammet; Akkemik, Ebru; Budak, Harun; Ciftci, Mehmet

Designing modulators of dimethylarginine dimethylaminohydrolase (DDAH): A focus on selectivity over arginase
pp. 24-28(5)
Authors: Kotthaus, Juerke; Schade, Dennis; Kotthaus, Joscha; Clement, Bernd

Biochemical characterization of an ectonucleotide pyrophosphatase/phosphodiesterase (E-NPP, E.C. 3.1.4.1) from rat cardiac soluble and microsomal fractions
pp. 29-36(8)
Authors: Pochmann, Daniela; Innocente, Adrine Maria; Buffon, Andréia; Freitas Sarkis, João José; Porciúncula, Lisiane De Oliveira

Evaluation of in vitro effects of some analgesic drugs on erythrocyte and recombinant carbonic anhydrase I and II
pp. 37-42(6)
Authors: Gökçe, Başşak; Gençer, Nahit; Arslan, Oktay; Turkoğğlu, Sumeyye Aydogan; Alper, Meltem; Köçkar, Feray

Synthesis and carbonic anhydrase inhibitory properties of novel bromophenols including natural products
pp. 43-50(8)
Authors: Balaydıın, Halis Türker; Soyut, Hakan; Ekinci, Deniz; Göksu, Süleyman; Beydemir, ŞŞükrü; Menzek, Abdullah; ŞŞahin, Ertan

Synthesis, antimicrobial activity and cytotoxicity of novel oxadiazole derivatives
pp. 51-57(7)
Authors: Kaplancikli, Zafer Asim; Altintop, Mehlika Dilek; Turan-Zitouni, Gulhan; Ozdemir, Ahmet; Ozic, Rasime; Akalıın, Gülşşen

Synthesis, characterization and biological studies of sulfonamide Schiff's bases and some of their metal derivatives
pp. 58-68(11)
Authors: Chohan, Zahid H.; Shad, Hazoor A.; Supuran, Claudiu T.

Synthesis and biological screening of some pyridine derivatives as anti-malarial agents
pp. 69-77(9)
Authors: Bekhit, Adnan A.; Hymete, Ariaya; Damtew, Ashenafi; Mohamed, Abdel Maaboud I.; Bekhit, Alaa El-Din A.

The phenylthiourea is a competitive inhibitor of the enzymatic oxidation of DOPA by phenoloxidase
pp. 78-83(6)
Authors: Ryazanova, Alexandra D.; Alekseev, Alexander A.; Slepneva, Irina A.

Thermal solvent-free synthesis of chromonyl chalcones, pyrazolines and their in vitro antibacterial, antifungal activities
pp. 84-91(8)
Authors: Siddiqui, Zeba N.; Praveen, Shagufta; Musthafa, T.N. Mohammed; Ahmad, Anis; Khan, Asad U.

Synthesis and biological evaluation of some novel sulfamoylphenyl-pyridazinone as anti-inflammatory agents (Part-II**)
pp. 92-96(5)
Authors: Bashir, Rafia; Yaseen, Shafiya; Ovais, Syed; Ahmad, Shamim; Hamid, Hinna; Alam, M.S.; Samim, Mohammad; Javed, Kalim

Carbonic anhydrase I and II inhibition with natural products: caffeine and piperine
pp. 97-100(4)
Authors: Sethi, Kalyan K.; Sahoo, Suvendu K.; Pichikala, Jayaprakash N.; Suresh, Padilam

Novel furfurylidene N-acylhydrazones derived from natural safrole: discovery of LASSBio-1215, a new potent antiplatelet prototype
pp. 101-109(9)
Authors: Rodrigues, Ana Paula C.; Costa, Luciana M.M.; Santos, Bruna L.R.; Maia, Rodolfo C.; Miranda, Ana L.P.; Barreiro, Eliezer J.; Fraga, Carlos A.M.

Synthesis and evaluation of anti-inflammatory, analgesic, ulcerogenic and lipid peroxidation properties of new 2-(4-isobutylphenyl)propanoic acid derivatives
pp. 110-116(7)
Authors: Raval, Jignesh Priyakant; Gandhi, Ankur Navinchandra; Akhaja, Tarunkumar Nanjibhai; Myangar, Kruti Navinbhai; Patel, Nilesh Hasmukhbhai

Chemical reactivity and antimicrobial activity of N-substituted maleimides
pp. 117-124(8)
Authors: Salewska, Natalia; Boros-Majewska, Joanna; ŁŁąącka, Izabela; Chylińńska, Katarzyna; Sabisz, Michałł; Milewski, Słławomir; Milewska, Maria J.

In vitro inhibition of polyphenol oxidase by some new diarylureas
pp. 125-131(7)
Authors: Demir, Dudu; Gençer, Nahit; Arslan, Oktay; Genç, Hayriye; Zengin, Mustafa

Rapid screening of enzyme inhibitors using Profiling of Enzyme-Metabolite Assay by HPLC (PREMA-HPLC)
pp. 132-137(6)
Authors: Vasantha, K.Y.; Murugesh, C.S.; Sattur, A.P.

A new approach to antiglaucoma drugs: carbonic anhydrase inhibitors with or without NO donating moieties. Mechanism of action and preliminary pharmacology
pp. 138-147(10)
Authors: Fabrizi, Francesca; Mincione, Francesco; Somma, Teresa; Scozzafava, Gabriele; Galassi, Fernando; Masini, Emanuela; Impagnatiello, Francesco; Supuran, Claudiu T.

α-Carbonic anhydrases are sulfatases with cyclic diol monosulfate esters
pp. 148-154(7)
Authors: Çavdar, Hüseyin; Ekinci, Deniz; Talaz, Oktay; Saraçoğğlu, Nurullah; ŞŞentürk, Murat; Supuran, Claudiu T.

Synthesis and biological evaluation of novel 6, 7-dimethoxy-3-(4-pyridyl)-2,3,3a,4-tetrahydroindeno[1,2-c]pyrazol-2-yl-4-substituted phenylmethanone/ethanone derivatives
pp. 155-159(5)
Authors: Ali, Mohamed Ashraf; Ismail, Rusli; Choon, Tan Soo; Elumalai, Manogaran; Kumar, Suresh; Osman, Hasnah; Govidasamy, Jeyabalan; Yadav, Rajesh; Yadav, Garima; Kour, Ravinder; Vyas, Swati

The crystal structure of protease Sapp1p from Candida parapsilosis in complex with the HIV protease inhibitor ritonavir
pp. 160-165(6)
Authors: Dostál, Jiřří; Brynda, Jiřří; Hrušková-Heidingsfeldová, Olga; Pachl, Petr; Pichová, Iva; ŘŘezáččová, Pavlína

Upcoming conferences of interest
pp. 166-166(1)
Author: Supuran, Claudiu T.