Journal of Enzyme Inhibition and Medicinal Chemistry

Efavirenz Mannich bases: Synthesis, anti-HIV and antitubercular activities
pp. 1-5(5)
Authors: Sriram, Dharmarajan; Banerjee, Debjani; Yogeeswari, Perumal

QSAR study of substituted 2-pyridinyl guanidines as selective urokinase-type plasminogen activator (uPA) inhibitors
pp. 6-13(8)
Authors: Karthikeyan, C.; Moorthy, N.S. Hari Narayana; Trivedi, Piyush

Inhibitory effects of flavonoids on aldehyde oxidase activity
pp. 14-21(8)
Authors: Pirouzpanah, Saeed; Hanaee, Jalal; Razavieh, Seyed-Vali; Rashidi, Mohammad-Reza

Alkaline phosphatase inhibition by vanadyl-β-diketone complexes: electron density effects
pp. 22-28(7)
Authors: Ziegler, Amanda; Florian, Jan; Ballicora, Miguel; Herlinger, Albert

Synthesis and characterization of some new 2(3H)-benzoxazolones with analgesic and antiinflammatory activities
pp. 29-37(9)
Authors: Gokhan-Kelekci, Nesrin; Koksal, Meric; Unuvar, Songul; Aktay, Goknur; Erdoğan, Hakki

His22 of TLXI plays a critical role in the inhibition of glycoside hydrolase family 11 xylanases
pp. 38-46(9)
Authors: Rombouts, Sigrid; Fierens, Ellen; Vandermarliere, Elien; Voet, Arnout; Gebruers, Kurt; Beaugrand, Johnny; Courtin, Christophe; Delcour, Jan; de Maeyer, Marc; Rabijns, Anja; Van Campenhout, Steven; Volckaert, Guido

New diterpenoid alkaloids from Aconitum heterophyllum Wall: Selective butyrylcholinestrase inhibitors
pp. 47-51(5)
Authors: Nisar, Muhammad; Ahmad, Manzoor; Wadood, Noreen; Lodhi, Muhammad Arif; Shaheen, Farzana; Choudhary, M. Iqbal

Unexpected formation of 3-chloro-1-hydroxy-2,6-diarylpiperidin-4-ones: Synthesis, antibacterial and antifungal activities
pp. 52-58(7)
Authors: Gopalakrishnan, M.; Thanusu, J.; Kanagarajan, V.; Govindaraju, R.

Isolation and characterization of a novel adenosine deaminase inhibitor, IADA-7, from Bacillus sp. J-89
pp. 59-64(6)
Authors: Lee, Gwang; Lee, Sang Seop; Kay, Kwang Yol; Kim, Dong Wan; Choi, Sangdun; Jun, Hong Ki

α-Glucosidase inhibitory activity of cyanidin-3-galactoside and synergistic effect with acarbose
pp. 65-69(5)
Authors: Adisakwattana, Sirichai; Charoenlertkul, Piyawan; Yibchok-anun, Sirintorn

Carbonic anhydrase inhibitors. Cloning, characterization and inhibition studies of the cytosolic isozyme III with anions
pp. 70-76(7)
Authors: Nishimori, Isao; Minakuchi, Tomoko; Onishi, Saburo; Vullo, Daniela; Cecchi, Alessandro; Scozzafava, Andrea; Supuran, Claudiu

Topological descriptors in modeling malonyl coenzyme A decarboxylase inhibitory activity: N-Alkyl-N-(1,1,1,3,3,3-hexafluoro-2-hydroxypropylphenyl)amide derivatives
pp. 77-85(9)
Authors: Singh, P.; Kumar, R.; Sharma, B. K.; Prabhakar, Y. S.

Modeling of vascular endothelial growth factor receptor 2 (VEGFR2) kinase inhibitory activity of 2-anilino-5-aryloxazoles using chemometric tools
pp. 86-93(8)
Authors: Sharma, B. K.; Sharma, S. K.; Singh, P.; Sharma, Susheela; Prabhakar, Y. S.

Topological descriptors in modelling antimalarial activity: N1-(7-chloro-4-quinolyl)-1,4-bis(3-aminopropyl)piperazine as prototype
pp. 94-104(11)
Authors: Deshpande, Shreekant; Solomon, V. Raja; Katti, Setu; Prabhakar, Yenamandra

Aluminium(III), chromium(III) and iron(III) complexes with 5-iodouracil and 5-iodouracil-histidine and their antitumour activity
pp. 105-110(6)
Authors: Singh, Vinod; Singh, Shweta; Narang, K. K.; Bhattacharya, D.

Kinetic properties and inhibition of the dimeric dUTPase-dUDPase from Campylobacter jejuni
pp. 111-116(6)
Authors: Musso-Buendia, Juan; Vidal, Antonio; Kasinthan, Ganasan; Nguyen, Corinne; Carrero-Lerida, Juana; Ruiz-perez, Luis; Wilson, Keith; Johansson, Nils Gunnar; Gilbert, Ian; Gonzalez-Pacanowska, Dolores

Synthesis and antitubercular activity of a series of hydrazone and nitrovinyl analogs derived from heterocyclic aldehydes
pp. 117-124(8)
Authors: Sonar, Vijayakumar; Crooks, Peter

A new Schiff base copper (II) complex derived from estrone and d-glucosamine: Synthesis, characterization and its interaction with DNA
pp. 125-130(6)
Authors: Yang, Xin-Bin; Wang, Li; Zhang, Ji; Zhang, Zhong-Wei; Lin, Hong-Hui; Zhou, Li-Hong; Yu, Xiao-Qi

Antiplasmodial activities of sesquiterpene lactone from Carpesium cernum
pp. 131-135(5)
Authors: Chung, Ill-Min; Moon, Hyung-In

Antidiabetic Effect of an Active Fraction Extracted from Dragon's Blood (Dracaena Cochinchinensis)
pp. 136-139(4)
Authors: Gu, Hui-Juan; Lv, Jing-Ci; Yong, Ke-Lan; Chen, Xu; Liu, Pei-Pei; Zhang, Xia-Bing

Synthesis, spectral characterization and microbiological studies of Co(II), Ni(II) and Cu(II) complexes with some novel 20-membered macrocyclic hydrazino-1,2,4-triazole Schiff bases
pp. 140-150(11)
Authors: Avaji, Prakash Gouda; Patil, Sangamesh Amarappa

In silico studies of urease inhibitors to explore ligand-enzyme interactions
pp. 151-156(6)
Authors: Ansari, Farzana Latif; Wadood, Abdul; Ullah, Ahsan; Iftikhar, Fatima; Ul-Haq, Zaheer

Computational neural network analysis of the affinity of N-n-alkylnicotinium salts for the α4β2* nicotinic acetylcholine receptor
pp. 157-168(12)
Authors: Zheng, Fang; Zheng, Guangrong; Deaciuc, A. Gabriela; Zhan, Chang-Guo; Dwoskin, Linda; Crooks, Peter

Synthesis of organometallic-based biologically active compounds: In vitro antibacterial, antifungal and cytotoxic properties of some sulfonamide incorporated ferrocences
pp. 169-175(7)
Author: Chohan, Zahid

4-phenyldiazenyl 2-(phenylimino methyl) phenols; synthesis and in-vitro biological evaluation as potential antibacterial agents
pp. 176-180(5)
Authors: Halve, Anand; Dubey, Pushp Kant; Kankoriya, Amit; Tiwari, Kiran

New N4-substituted piperazine naphthamide derivatives as BACE-1 inhibitors
pp. 181-187(7)
Authors: Laras, Y.; Garino, C.; Dessolin, J.; Weck, C.; Moret, V.; Rolland, A.; Kraus, J. -L.

Quinic acid derivatives from Saussurea triangulata attenuates glutamate-induced neurotoxicity in primary cultured rat cortical cells
pp. 188-191(4)
Authors: Chung, Ill-Min; Kim, Min-Young; Park, Won-Hwan; Moon, Hyung-In

In vitro antifungal and antibacterial activities of extracts of Galium tricornutum subsp. longipedunculatum
pp. 192-196(5)
Authors: Khaliq Jan, Abdul; Raza Shah, Muhammad; Anis, Itrat; Khan Marwat, Inamullah

Synthesis, characterization and antimicrobial activities of some mixed ligand complexes of Co(II) with thiosemicarbazones and N-protected amino acids
pp. 197-204(8)
Authors: Sharma, Renu; Nagar, Meena; Agarwal, Manoj; Sharma, Hemant

Predictive QSAR modeling of CCR5 antagonist piperidine derivatives using chemometric tools
pp. 205-223(19)
Authors: Roy, Kunal; Mandal, Asim Sattwa

Antibacterial, antifungal, insecticidal, cytotoxicity and phytotoxicity studies on Indigofera gerardiana
pp. 224-229(6)
Authors: Nisar, Muhammad; Tariq, Shafiq Ahmad; Marwat, Inamullah Khan; Shah, Muhammad Raza; Khan, Ihsan Ali

Chemical constituents isolated from Polygala japonica leaves and their inhibitory effect on nitric oxide production in vitro
pp. 230-233(4)
Authors: Kim, Seung Hyun; Jang, Sin-Duk; Lee, Ki Yong; Sung, Sang Hyun; Kim, Young Choong

The leaf extract of Siberian Crabapple (Malus baccata (Linn.) Borkh) contains potential fatty acid synthase inhibitors
pp. 234-240(7)
Authors: Wei, Xiang; Zhao, Ran; Sun, Ying-Hui; Cong, Jian-Ping; Meng, Fan-Guo; Zhou, Hai-Meng

The strand transfer oligonucleotide inhibitors of HIV-integrase
pp. 241-246(6)
Authors: Snasel, Jan; Rosenberg, Ivan; Paces, Ondrej; Pichova, Iva

In vivo antiplasmodial activity of 11(13)-dehydroivaxillin from Carpesium ceruum
pp. 247-250(4)
Authors: Kim, Jong-Jin; Chung, Ill-Min; Jung, Jae-Chul; Kim, Min-Young; Moon, Hyung-In

Inhibitory effects of Cefazolin and Cefodizime on the activity of mushroom tyrosinase
pp. 251-256(6)
Authors: Zhuang, Jiang-Xing; Li, Wen-Gang; Qiu, Ling; Zhong, Xue; Zhou, Jing-Jing; Chen, Qing-Xi

Protein glycation inhibitory activities of Lawsonia inermis and its active principles
pp. 257-261(5)
Authors: Sultana, Nighat; Choudhary, Muhammed Iqbal; Khan, Ambrin

QSAR study on dual SET and NET reuptake inhibitors: An insight into the structural requirement for antidepressant activity
pp. 262-271(10)
Author: Dessalew, Nigus

CoMFA and CoMSIA 3D-QSAR analysis on hydroxamic acid derivatives as urease inhibitors
pp. 272-278(7)
Authors: Ul-Haq, Zaheer-; Wadood, Abdul; Uddin, Reaz

Inhibition of rat liver cathepsins B and L by the peptide aldehyde benzyloxycarbonyl-leucyl-leucyl-leucinal and its analogues
pp. 279-286(8)
Authors: Ito, Hisashi; Watanabe, Masafumi; Kim, Yong-Tae; Takahashi, Kenji

Green tea catechins in chemoprevention of cancer: A molecular docking investigation into their interaction with glutathione S-transferase (GST P1-1)
pp. 287-295(9)
Authors: Artali, Roberto; Beretta, Giangiacomo; Morazzoni, Paolo; Bombardelli, Ezio; Meneghetti, Fiorella

Synthesis of some pyrazolyl benzenesulfonamide derivatives as dual anti-inflammatory antimicrobial agents
pp. 296-309(14)
Authors: Bekhit, Adnan; Ashour, Hayam; Bekhit, Alaa El-Din; Abdel-Rahman, Hamdy; Bekhit, Salma

Corrigendum
pp. 310-314(5)
Authors: Bekhit, Adnan; Ashour, Hayam; Bekhit, Alaa El-Din; Abdel-Rahman, Hamdy; Bekhit, Salma