Insulinomimetic bis(maltolato)zinc(II) Complex: Blood Glucose Normalizing Effect in KK-Ay Mice with Type 2 Diabetes Mellitus
Authors: Yoshikawa Y.1; Ueda E.1; Miyake H.1; Sakurai H.2; Kojima Y.1
Source: Biochemical and Biophysical Research Communications, Volume 281, Number 5, March 2001 , pp. 1190-1193(4)
Publisher: Academic Press
Abstract:
High blood glucose levels of KK-Ay mice with type 2 diabetes mellitus were normalized by daily intraperitoneal (ip) administration of a zinc(II) complex, bis(maltolato)zinc(II) (Zn(Mal)2) with a Zn(O4) coordination mode, following the finding of strong in vitro insulinomimetic activity in isolated rat adipocytes treated with epinephrine in terms of the inhibition of free fatty acid release. The blood glucose level was maintained in the normal range during administration of the Zn(Mal)2 complex for 14 days and improvements in the glucose tolerance were confirmed by an oral glucose tolerance test. Copyright 2001 Academic Press.
Keywords: zinc complex; KK-Ay mice; blood glucose normalizing effect
Language: English
Document Type: Research article
Affiliations: 1: Graduate School of Science, Osaka City University, 3-3-138 Sugimoto, Sumiyoshi-ku, Osaka, 558-8585, Japan 2: Department of Analytical and Bioinorganic Chemistry, Kyoto Pharmaceutical University, 5 Nakauchi-cho, Misasagi, Yamashina-ku, Kyoto, 607-8414, Japan

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